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1

Studies on the mechanism of action of win 49596: A steroidal androgen receptor antagonist

Richard C. Winneker, Margaret M. Wagner, Frederick H. Batzold

Journal:

Journal of Steroid Biochemistry

Year:

1989

Language:

english

File:

PDF, 709 KB

english, 1989

2

Endocrine profile of win 49596 in the rat: A novel androgen receptor antagonist

Ben W. Snyder, Richard C. Winneker, Frederick H. Batzold

Journal:

Journal of Steroid Biochemistry

Year:

1989

Language:

english

File:

PDF, 684 KB

english, 1989

3

In vitro characterization of trimegestone: a new potent and selective progestin

Zhiming Zhang, Scott G Lundeen, Yuan Zhu, Jeffrey M Carver, Richard C Winneker

Journal:

Year:

2000

Language:

english

File:

PDF, 594 KB

english, 2000

4

The preclinical biology of a new potent and selective progestin: trimegestone

Richard C Winneker, Daniel Bitran, Zhiming Zhang

Journal:

Year:

2003

Language:

english

File:

PDF, 274 KB

english, 2003

5

Rat uterine complement C3 expression as a model for progesterone receptor modulators: characterization of the new progestin trimegestone

Scott G Lundeen, Zhiming Zhang, Yuan Zhu, Jeffrey M Carver, Richard C Winneker

Journal:

The Journal of Steroid Biochemistry and Molecular Biology

Year:

2001

Language:

english

File:

PDF, 268 KB

english, 2001

6

Antiandrogenic steroidal sulfonylpyrazoles

Christiansen, Robert G., Bell, Malcolm R., D'Ambra, Thomas E., Mallamo, John P., Herrmann, John L., Ackerman, James H., Opalka, Chester J., Kullnig, Rudolph K., Winneker, Richard C.

Journal:

Journal of Medicinal Chemistry

Year:

1990

Language:

english

File:

PDF, 1.77 MB

english, 1990

7

ChemInform Abstract: Potent Nonsteroidal Progesterone Receptor Agonists: Synthesis and SAR Study of 6-Aryl Benzoxazines.

Puwen Zhang, Eugene A. Terefenko, Andrew Fensome, Zhiming Zhang, Yuan Zhu, Jeffrey Cohen, Richard Winneker, Jay Wrobel, John Yardley

Journal:

Year:

2002

Language:

english

File:

PDF, 31 KB

english, 2002

8

Effects of the steroidal antiandrogen win 49596 on fertility and sex accessory tissue growth in the rat

Frederick H. Batzold, Richard C. Winneker, Ben W. Snyder, Jerry R. Reel

Journal:

Drug Development Research

Year:

1990

Language:

english

File:

PDF, 431 KB

english, 1990

9

5-(3-Cyclopentyl-2-thioxo-2,3-dihydro-1H-benzimidazol-5-yl)-1-methyl-1H-pyrrole-2-carbonitrile: A novel, highly potent, selective, and orally active non-steroidal progesterone receptor agonist

Puwen Zhang, Eugene Terefenko, Jeffrey Kern, Andrew Fensome, Eugene Trybulski, Ray Unwalla, Jay Wrobel, Susan Lockhead, Yuan Zhu, Jeffrey Cohen, Margaret LaCava, Richard C. Winneker, Zhiming Zhang

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 403 KB

english, 2007

10

7-Aryl 1,5-dihydro-benzo[e][1,4]oxazepin-2-ones and analogs as non-steroidal progesterone receptor antagonists

Puwen Zhang, Jeffrey C. Kern, Eugene A. Terefenko, Andrew Fensome, Ray Unwalla, Zhiming Zhang, Jeffrey Cohen, Thomas J. Berrodin, Matthew R. Yudt, Richard C. Winneker, Jay Wrobel

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 450 KB

english, 2008

11

SAR studies of 6-aryl-1,3-dihydrobenzimidazol-2-ones as progesterone receptor antagonists

Eugene A. Terefenko, Jeffrey Kern, Andrew Fensome, Jay Wrobel, Yuan Zhu, Jeffrey Cohen, Richard Winneker, Zhiming Zhang, Puwen Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 166 KB

english, 2005

12

SAR studies of 6-(arylamino)-4,4-disubstituted-1-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-ones as progesterone receptor antagonists

Jeffrey C. Kern, Eugene A. Terefenko, Andrew Fensome, Ray Unwallla, Jay Wrobel, Yuan Zhu, Jeffrey Cohen, Richard Winneker, Zhiming Zhang, Puwen Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 138 KB

english, 2007

13

1,5-Dihydro-benzo[e][1,4]oxazepin-2(1H)-ones containing a 7-(5′-cyanopyrrol-2-yl) group as nonsteroidal progesterone receptor modulators

Jeffrey C. Kern, Eugene A. Terefenko, Andrew Fensome, Ray Unwalla, Jay Wrobel, Jeffrey Cohen, Yuan Zhu, Thomas J. Berrodin, Matthew R. Yudt, Richard C. Winneker, Zhiming Zhang, Puwen Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 168 KB

english, 2008

14

5-Aryl indanones and derivatives as non-steroidal progesterone receptor modulators

Jeffrey C. Kern, Eugene Terefenko, Eugene Trybulski, Thomas J. Berrodin, Jeffrey Cohen, Richard C. Winneker, Matthew R. Yudt, Zhiming Zhang, Yuan Zhu, Puwen Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 242 KB

english, 2009

15

1-Methyl-1H-pyrrole-2-carbonitrile containing tetrahydronaphthalene derivatives as non-steroidal progesterone receptor antagonists

Jeffrey C. Kern, Eugene Terefenko, Eugene Trybulski, Thomas J. Berrodin, Jeffrey Cohen, Richard C. Winneker, Matthew R. Yudt, Zhiming Zhang, Yuan Zhu, Puwen Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 466 KB

english, 2010

16

New progesterone receptor antagonists: 3,3-disubstituted-5-aryloxindoles

Andrew Fensome, Reinhold Bender, Jeffrey Cohen, Mark A. Collins, Valerie A. Mackner, Lori L. Miller, John W. Ullrich, Richard Winneker, Jay Wrobel, Puwen Zhang, Zhiming Zhang, Yuan Zhu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 112 KB

english, 2002

17

Novel 5-aryl-1,3-dihydro-indole-2-thiones: potent, orally active progesterone receptor agonists

Andrew Fensome, Marci Koko, Jay Wrobel, Puwen Zhang, Zhiming Zhang, Jeffrey Cohen, Scott Lundeen, Kelly Rudnick, Yuan Zhu, Richard Winneker

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 192 KB

english, 2003

18

Novel 6-aryl-1,4-dihydrobenzo[d]oxazine-2-thiones as potent, selective, and orally active nonsteroidal progesterone receptor agonists

Puwen Zhang, Eugene A. Terefenko, Andrew Fensome, Jay Wrobel, Richard Winneker, Zhiming Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 198 KB

english, 2003

19

Molecular analysis of the vaginal response to estrogens in the ovariectomized rat and postmenopausal woman

Scott A Jelinsky, Sung E Choe, Judy S Crabtree, Monette M Cotreau, Ewa Wilson, Kathryn Saraf, Andrew J Dorner, Eugene L Brown, Bryan J Peano, Xiaochun Zhang, Richard C Winneker, Heather A Harris

Journal:

BMC Medical Genomics

Year:

2008

Language:

english

File:

PDF, 1.51 MB

english, 2008

20

Novel pyrrole-containing progesterone receptor modulators

Mark A Collins, Valerie Hudak, Reinhold Bender, Andrew Fensome, Puwen Zhang, Lori Miller, Richard C Winneker, Zhiming Zhang, Yuan Zhu, Jeffrey Cohen, Rayomond J Unwalla, Jay Wrobel

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2004

Language:

english

File:

PDF, 282 KB

english, 2004

21

Synthesis and androgen receptor affisity of steroidal methylsulfonylforans and a menthylsulfonylthiophene

Virendra Kumar, Sol J. Daum, Malcolm R. Bell, Michael A. Alexander, Robert G. Christiansen, James H. Ackerman, Michael E. Krolski, Carry M. Pilling, John L. Herrmann Jr., Richard C. Winneker, Margaret

Journal:

Year:

1991

Language:

english

File:

PDF, 694 KB

english, 1991

22

Potent nonsteroidal progesterone receptor agonists: Synthesis and SAR study of 6-aryl benzoxazines

Puwen Zhang, Eugene A. Terefenko, Andrew Fensome, Zhiming Zhang, Yuan Zhu, Jeffrey Cohen, Richard Winneker, Jay Wrobel, John Yardley

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 120 KB

english, 2002

23

The angiogenic factor Cyr61 is induced by the progestin R5020 and is necessary for mammary adenocarcinoma cell growth

Deepak Sampath, Richard C. Winneker, Zhiming Zhang

Journal:

Endocrine (Springer)

Year:

2002

Language:

english

File:

PDF, 382 KB

english, 2002

24

10.1021/ja01255a030

Roblin, Richard O., Winnek, Philip S., English, Jackson P.

Journal:

Journal of the American Chemical Society

Year:

1942

Language:

english

File:

PDF, 457 KB

english, 1942

25

Novel progesterone receptor modulators with gene selective and context-dependent partial agonism

Thomas J. Berrodin, Scott A. Jelinsky, Nilsa Graciani, John A. Butera, Zhiming Zhang, Sunil Nagpal, Richard C. Winneker, Matthew R. Yudt

Journal:

Biochemical Pharmacology

Year:

2009

Language:

english

File:

PDF, 1.16 MB

english, 2009

26

TNF-α and 9-cis-Retinoic Acid Synergistically Induce ICAM-1 Expression: Evidence for Interaction of Retinoid Receptors with NF-κB

Christopher C. Chadwick, Lucinda J. Shaw, Richard C. Winneker

Journal:

Experimental Cell Research

Year:

1998

Language:

english

File:

PDF, 178 KB

english, 1998

27

Differing pharmacological activities of thiazolidinone analogs at the FSH receptor

Brian J. Arey, Stephen D. Yanofsky, M. Claudia Pérez, Christopher P. Holmes, Jay Wrobel, Ariamala Gopalsamy, Panayiotis E. Stevis, Francisco J. López, Richard C. Winneker

Journal:

Biochemical and Biophysical Research Communications

Year:

2008

Language:

english

File:

PDF, 362 KB

english, 2008

28

Identification of novel estrogen receptor α antagonists

Dalei Shao, Thomas J Berrodin, Eric Manas, Diane Hauze, Robert Powers, Ashok Bapat, Daniel Gonder, Richard C Winneker, Donald E Frail

Journal:

The Journal of Steroid Biochemistry and Molecular Biology

Year:

2004

Language:

english

File:

PDF, 369 KB

english, 2004

29

Differential effects of estrogens and progestins on the anticoagulant tissue factor pathway inhibitor in the rat

Rebecca A. Shirk, Zhiming Zhang, Richard C. Winneker

Journal:

The Journal of Steroid Biochemistry and Molecular Biology

Year:

2005

Language:

english

File:

PDF, 209 KB

english, 2005

30

Quantitative analysis of gene regulation by seven clinically relevant progestins suggests a highly similar mechanism of action through progesterone receptors in T47D breast cancer cells

Jeffrey D. Bray, Scott Jelinsky, Radhika Ghatge, Jenifer A. Bray, Christopher Tunkey, Kathryn Saraf, Britta M. Jacobsen, Jennifer K. Richer, Eugene L. Brown, Richard C. Winneker, Kathryn B. Horwitz, C

Journal:

The Journal of Steroid Biochemistry and Molecular Biology

Year:

2005

Language:

english

File:

PDF, 648 KB

english, 2005

31

Development of a mouse model of mammary gland versus uterus tissue selectivity using estrogen- and progesterone-regulated gene markers

Judy S. Crabtree, Xiaochun Zhang, Bryan J. Peano, Zhiming Zhang, Richard C. Winneker, Heather A. Harris

Journal:

The Journal of Steroid Biochemistry and Molecular Biology

Year:

2006

Language:

english

File:

PDF, 1.12 MB

english, 2006

32

Activity of three selective estrogen receptor modulators on hormone-dependent responses in the mouse uterus and mammary gland

Judy S. Crabtree, Bryan J. Peano, Xiaochun Zhang, Barry S. Komm, Richard C. Winneker, Heather A. Harris

Journal:

Molecular and Cellular Endocrinology

Year:

2008

Language:

english

File:

PDF, 953 KB

english, 2008

33

A new generation of progesterone receptor modulators

Richard C. Winneker, Andrew Fensome, Puwen Zhang, Matthew R. Yudt, Casey C. McComas, Rayomond J. Unwalla

Journal:

Year:

2008

Language:

english

File:

PDF, 702 KB

english, 2008

34

Regulation of gene expression by PRA-910, a novel progesterone receptor modulator, in T47D cells

Jeffrey D Bray, Zhiming Zhang, Richard C Winneker, C.Richard Lyttle

Journal:

Year:

2003

Language:

english

File:

PDF, 132 KB

english, 2003

35

The effect of estrogens and antiestrogens in a rat model for hot flush

Istvan Merchenthaler, Judith M. Funkhouser, Jeffrey M. Carver, Scott G. Lundeen, Krishnendu Ghosh, Richard C. Winneker

Journal:

Year:

1998

Language:

english

File:

PDF, 246 KB

english, 1998

36

Antiandrogenic steroidal sulfonyl heterocycles. Utility of electrostatic complementarity in defining bioisosteric sulfonyl heterocycles

Mallamo, John P., Pilling, Garry M., Wetzel, Joseph R., Kowalczyk, Paul J., Bell, Malcolm R., Kullnig, Rudolph K., Batzold, Frederick H., Juniewicz, Paul E., Winneker, Richard C., Luss, Henry R.

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 2.07 MB

english, 1992

37

Glucocorticoid/Antiinflammatory activities of nonsteroidal phenylpyrazoles in the rat

H. Philip Schane, Homer R. Harding, Malcolm R. Bell, V. Daniel Castracane, Richard C. Winneker, Ben W. Snyder

Journal:

Year:

1985

Language:

english

File:

PDF, 646 KB

english, 1985

38

Identification of genes involved in follicular development by transcription gene profiling of ovaries from 5 and 15-day old mice

Maria Claudia Perez, Richard Craig Winneker

Journal:

Fertility and Sterility

Year:

2002

Language:

english

File:

PDF, 31 KB

english, 2002

39

The interaction of nivazol with the glucocorticoid receptor from rat and rhesus monkey target tissues

Richard C. Winneker, Margaret M. Russell, Christine K. Might, H. Philip Schane

Journal:

Year:

1984

Language:

english

File:

PDF, 545 KB

english, 1984

40

Chemotherapy. II. Some Sulfanilamido Heterocycles 1

Roblin, Richard O., Williams, James H., Winnek, Philip S., English, Jackson P.

Journal:

Journal of the American Chemical Society

Year:

1940

Language:

english

File:

PDF, 425 KB

english, 1940

41

Non-steroidal glucocorticoid-like substances: receptor binding and in vivo activity

Kumar, Virendra, Bell, Malcolm R., Wetzel, Joseph R., Herrmann, John L., McGarry, Ruthann, Schane, H. Phillip, Winneker, Richard C., Snyder, Ben W., Anzalone, Anthony J.

Journal:

Journal of Medicinal Chemistry

Year:

1993

Language:

english

File:

PDF, 825 KB

english, 1993

42

Alleviation of Thermoregulatory Dysfunction with the New Serotonin and Norepinephrine Reuptake Inhibitor Desvenlafaxine Succinate in Ovariectomized Rodent Models

Deecher, Darlene C., Alfinito, Peter D., Leventhal, Liza, Cosmi, Scott, Johnston, Grace H., Merchenthaler, Istvan, Winneker, Richard

Journal:

Year:

2007

Language:

english

File:

PDF, 281 KB

english, 2007

43

Novel progesterone receptor modulators: 4-Aryl-phenylsulfonamides

McComas, Casey, Cohen, Jeffrey, Huselton, Christine, Marella, Michael, Melenski, Edward, Mugford, Cheryl, Slayden, Ov, Winneker, Richard, Wrobel, Jay, Yudt, Matthew R., Fensome, Andrew

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 703 KB

english, 2012

44

A Mouse Model of Androgenetic Alopecia

Crabtree, Judy S., Kilbourne, Edward J., Peano, Bryan J., Chippari, Susan, Kenney, Thomas, McNally, Christopher, Wang, Wei, Harris, Heather A., Winneker, Richard C., Nagpal, Sunil, Thompson, Catherine

Journal:

Year:

2010

Language:

english

File:

PDF, 397 KB

english, 2010

45

Chemotherapy. I. Substituted Sulfanilamidopyridines 1

Roblin, Richard O., Winnek, Philip S.

Journal:

Journal of the American Chemical Society

Year:

1940

Language:

english

File:

PDF, 449 KB

english, 1940

46

A novel, nonsteroidal inhibitor of androgen binding to the rat androgen binding protein: diethyl [[[3-(2,6-dimethyl-4-pyridinyl)-4-fluorophenyl]amino]methylene]propanedioate

Winneker, Richard C., Wagner, Margaret M., Singh, Baldev

Journal:

Journal of Medicinal Chemistry

Year:

1990

Language:

english

File:

PDF, 570 KB

english, 1990

47

6-Aryl-1,4-dihydro-benzo[ d ][1,3]oxazin- 2-ones: A Novel Class of Potent, Selective, and Orally Active Nonsteroidal Progesterone Receptor Antagonists †

Zhang, Puwen, Terefenko, Eugene A., Fensome, Andrew, Wrobel, Jay, Winneker, Richard, Lundeen, Scott, Marschke, Keith B., Zhang, Zhiming

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 61 KB

english, 2002

48

Studies in Chemotherapy. V. Sulfanilylcyanamide and Related Compounds 1

Winnek, Philip S., Anderson, George W., Marson, Harry W., Faith, H. Eldridge, Roblin, Richard O.

Journal:

Journal of the American Chemical Society

Year:

1942

Language:

english

File:

PDF, 459 KB

english, 1942

49

Studies in Chemotherapy. VI. Sulfanilamido Heterocycles 1

Anderson, George W., Faith, H. Eldridge, Marson, Harry W., Winnek, Philip S., Roblin, Richard O.

Journal:

Journal of the American Chemical Society

Year:

1942

Language:

english

File:

PDF, 472 KB

english, 1942

50

Non-steroidal progesterone receptor modulators

Zhang, Puwen, Fensome, Andrew, Wrobel, Jay, Winneker, Richard, Zhang, Zhiming

Journal:

Expert Opinion on Therapeutic Patents

Year:

2003

Language:

english

File:

PDF, 146 KB

english, 2003